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Sugammadex

Reversal of rocuronium/vecuronium neuromuscular blockade

Indications

  • Reversal of rocuronium/vecuronium neuromuscular blockade

Adult dosing

  • immediate reversal: dose: 16; unit: mg/kg; route: IV; weightBased: true; maxDose: 3200; maxDoseAbsolute: true; routine reversal: dose: 4; unit: mg/kg; route: IV; weightBased: true; maxDose: 800; maxDoseAbsolute: true

Pediatric dosing

  • routine reversal: dose: 2; unit: mg/kg; route: IV; weightBased: true; maxDose: 200; maxDoseAbsolute: true; immediate reversal: dose: 16; unit: mg/kg; route: IV; weightBased: true; maxDose: 1120; maxDoseAbsolute: true

Contraindications

  • Hypersensitivity to sugammadex

Clinical pearls

  • Use 16 mg/kg for immediate "cannot intubate, cannot ventilate" reversal of rocuronium
  • Encapsulates rocuronium — rendering it inactive; does not work for succinylcholine
  • May reduce efficacy of hormonal contraceptives — counsel patients
  • Onset faster and more predictable than neostigmine

Source and review

  • Tintinalli's Emergency Medicine, 9th ed.. Last reviewed: 2024-11-01